Substance Structure:
Individual bifunctional chemical compound of the carboxamide class, combining aminomethylisoxazole and nicotinic acid residues via a direct bond.
Mechanism of Action:
Increased lipophilicity and masking of the polar zwitterion to overcome the BBB via passive transmembrane diffusion without degradation in the GI tract.
Bioeffect and Properties:
Release of active components within the CNS. Synergistic anxiolytic, sedative, and cerebral vasodilating effects.
Commercialization Type:
Commercialization Type: B2B Bulk Ingredient for encapsulation. Supply of high-purity substance for creating ready-to-use formulation blends.
Technological Tools:
Targeted organic synthesis of bifunctional compounds, covalent binding of active components, analytical control of BBB permeability.
Msc-NH-Nic
TARGETED MOLECULAR STRUCTURE WITH IMPROVED BBB PERMEABILITY